Preview

Drug development & registration

Advanced search

Search


Order results by:     
 
Issue Title
 
Vol 13, No 1 (2024) Phase I Pharmacokinetics Study of Oral Administration of Esperavir® (INN: Molnupiravir) (LLC "PROMOMED RUS", Russia) Abstract  PDF (Rus)  similar documents
T. N. Komarov, N. S. Bagaeva, K. K. Karnakova, K. Ya. Zaslavskaya, P. A. Bely, I. E. Shohin
"... исследования является изучение фармакокинетики препарата Эсперавир®, капсулы 200 мг (АО «Биохимик», держатель ..."
 
Vol 13, No 4 (2024) Liposomes – metabolically active drug transport systems: visualization and pharmacokinetic. Part 2 (review) Abstract  PDF (Rus)  similar documents
O. N. Pozharitskaya, Yu. M. Kozur, S. S. Osochuk, E. V. Flisyuk, I. E. Smekhova, S. D. Malkov, K. O. Zarifi, I. A. Titovich, E. K. Krasova, A. N. Shikov
"... Введение. Во второй части обзора рассмотрены вопросы визуализации, фармакокинетики и ..."
 
Vol 9, No 4 (2020) Pharmacokinetic and Bioequivalence Study of Telzap AM® (Telmisartan/amlodipine Fixed-dose Combination) and Coadministered Mikardis® (Telmisartan) and Norvask® (Amlodipine) in Healthy Subjects Abstract  PDF (Rus)  similar documents
V. Kubesh, A. L. Khokhlov, A. M. Shitova, Yu. A. Dzhurko, V. I. Kazey, A. A. Khokhlov, A. E. Miroshnikov, O. V. Lebedeva, I. K. Klaus, A. V. Zyatenkov
"... сравнительное изучение фармакокинетики и подтверждение биоэквивалентности двухкомпонентного препарата Телзап® АМ ..."
 
Vol 12, No 1 (2023) Pharmacokinetic and Bioequivalence Study of the Two-component Drug Product "Ezetimibe + rosuvastatin" (JSC "Sanofi-aventis group", Russia): Resuts and Experience with the Use of Enzymatic Hydrolysis in the Analysis of Samples Abstract  PDF (Rus)  similar documents
A. L. Khokhlov, D. Yu. Grebenkin, E. K. Faeva, V. I. Kazey, A. A. Khokhlov, A. E. Miroshnikov, O. V. Lebedeva
"... добровольцев. Для оценки фармакокинетики общего эзетимиба использовали ферментативный гидролиз, что послужило ..."
 
Vol 13, No 1 (2024) Phase I Pharmacokinetics Study of Drug Areplivir® Zinc (INN: Favipiravir + Zinc Gluconate) (LLC "PROMOMED RUS", Russia) Abstract  PDF (Rus)  similar documents
T. N. Komarov, N. S. Bagaeva, K. K. Karnakova, O. A. Archakova, D. S. Shchelgacheva, V. S. Shcherbakova, K. Ya. Zaslavskaya, P. A. Bely, A. V. Taganov, I. E. Shohin
"... является изучение фармакокинетики препарата Арепливир® Цинк (МНН: фавипиравир + глюконат цинка), 200 + 70 ..."
 
Vol 13, No 1 (2024) Reciprocal Impact of Molnupiravir and Favipiravir Monocomponents of the Combination Drug on Each Other's Pharmacokinetics in a Phase I Clinical Trial Abstract  PDF (Eng)  similar documents
T. N. Komarov, K. K. Karnakova, N. S. Bagaeva, O. A. Archakova, M. O. Popova, V. S. Shcherbakova, K. Ya. Zaslavskaya, P. A. Bely, I. E. Shohin
"... "PROMOMED RUS", Russia). The plasma concentration of β-D-N4-hydroxycytidine (NHC), the active metabolite ..."
 
Vol 12, No 3 (2023) A Double-blind Randomized Comparative Phase I Study to Assess Biosimilarity and Immunogenicity of "Trastuzumab" (LLC "Mabscale", Russia) and Herceptin® (F. Hoffmann-La Roche Ltd., Switzerland) in Healthy Volunteers Abstract  PDF (Rus)  similar documents
M. A. Kolganova, E. E. Beketov, V. V. Pisarev, A. V. Ivanov, S. V. Vasiliev, I. E. Shokhin
"... сравнительного клинического исследования фармакокинетики и безопасности препаратов трастузумаба с участием ..."
 
Online First Physiologically-based pharmacokinetic modeling: past, present and future (review) Abstract  PDF (Rus)  similar documents
N. S. Bagaeva, E. I. Evtyukhina, D. S. Shchelgacheva, M. O. Popova, O. A. Archakova, T. N. Komarov, A. N. Marchenko, E. A. Malashenko, I. E. Shohin
"... Введение. Физиологически обоснованное моделирование фармакокинетики представляет собой метод ..."
 
Vol 11, No 1 (2022) Pharmacokinetics Study of the Long-acting Antiarrhythmic Drug of Lappaconitine Hydrobromide (Allaforte®, JSC "Pharmcenter VILAR", Russia) Abstract  PDF (Eng)  similar documents
O. A. Archakova, N. S. Bagaeva, T. N. Komarov, A. V. Rogov, D. S. Shchelgacheva, A. V. Suvorova, P. K. Karnakova, P. A. Karpova, I. E. Shohin
"... and methods. Concentration of lappaconitine and its active metabolite N-desacetyllappaconitine in human plasma ..."
 
Vol 12, No 2 (2023) Phase I Pharmacokinetics Study of Drug for Infusion «Areplivir» (INN: Favipiravir) (LLC "PROMOMED RUS", Russia) Abstract  PDF (Rus)  similar documents
T. N. Komarov, N. S. Bagaeva, K. K. Karnakova, I. E. Shohin, K. Ya. Zaslavskaya, P. A. Bely
"... исследования является изучение фармакокинетики препарата «Арепливир», лиофилизат для приготовления концентрата ..."
 
Vol 11, No 2 (2022) Phase I Pharmacokinetics Study of Drug «COVID-globulin» (Specific Human Immunoglobulin Against COVID-19) Abstract  PDF (Eng)  similar documents
T. I. Smolyanova, N. S. Bagaeva, M. A. Kolganova, I. E. Shohin, A. M. Nikolaeva, T. V. Vyaznikova, A. A. Pankratova, E. A. Bykova
"... является изучение фармакокинетики препарата «КОВИД-глобулин» (специфический иммуноглобулин человека против ..."
 
Vol 10, No 3 (2021) Determination of Lappaconitin, Diterpene Alkaloide Obtained from Plants Aconitum leucostomum, and its Active Metabolite N-desacetyllappaconitin in Human Plasma and Blood Abstract  PDF (Eng)  similar documents
O. A. Archakova, T. N. Komarov, A. V. Rogov, D. S. Shchelgacheva, A. A. Aleshina, N. S. Bagaeva, I. E. Shohin
"... pharmacologically active substances, but N-desacetyllappaconitine is the most effective. Drugs based ..."
 
Vol 10, No 4 (2021) Simultaneous Determination of Candesartan and Hydrochlorothiazide in Human Plasma by HPLC-MS/MS Abstract  PDF (Rus)  similar documents
P. K. Karnakova, T. N. Komarov, O. A. Archakova, D. S. Shchelgacheva, A. A. Aleshina, N. S. Bagaeva, P. A. Karpova, I. E. Shohin
"... . A., Shchelgacheva D. S., Aleshina A. A., Bagaeva N. S., Karpova P. A., Shohin I. E., 2021 ..."
 
Vol 11, No 2 (2022) Development and Validation of a Method for Determining Deferasirox in Human Blood Plasma by HPLC-UV Abstract  PDF (Eng)  similar documents
P. A. Karpova, T. N. Komarov, O. A. Archakova, D. S. Shchelgacheva, A. V. Suvorova, N. S. Bagaeva, P. K. Karnakova, I. E. Shohin
"... детектированием (ВЭЖХ-УФ) для дальнейшего исследования фармакокинетики и биоэквивалентности лекарственных ..."
 
Vol 13, No 2 (2024) Development and validation of a high-performance liquid chromatography with tandem mass spectrometry method for quantification of tofacitinib in human plasma Abstract  PDF (Eng)  similar documents
E. S. Vetrova, P. K. Karnakova, N. S. Bagaeva, K. K. Karnakova, M. O. Popova, A. A. Popova, O. A. Archakova, T. N. Komarov, I. E. Shohin
 
Vol 12, No 3 (2023) Determination of Favipiravir in Human Blood Plasma by HPLC-MS/MS Abstract  PDF (Eng)  similar documents
T. N. Komarov, P. A. Karpova, O. A. Archakova, D. S. Shchelgacheva, P. K. Karnakova, N. S. Bagaeva, K. Ya. Zaslavskaya, P. A. Bely, I. E. Shohin
"... with tandem mass-selective detection (HPLC-MS/MS) in order to study the pharmacokinetics of β-D-N4 ..."
 
Vol 8, No 3 (2019) A Comparative Parallel Study of Pharmacokinetics and Immunogenicity Following Single Intravenous Administration of Bevacizumab Biosimilar RPH-001 (Manufactured by R-Pharm Group, Russia) and Avastin® (Manufactured by F. Hoffmann-La Roche Ltd., Switzerland) in Healthy Male Volunteers Abstract  PDF (Rus)  similar documents
M. A. Kolganova, N. S. Bagaeva, Yu. V. Medvedev, I. E. Shohin, A. V. Demchinskaya, T. N. Palkina, D. A. Salazanov, G. E. Konopleva, M. S. Sheremeteva, Sh. Z. Archuadze, Ya. V. Lavrovsky, A. Yu. Savchenko, M. Yu. Samsonov
"... фазы для оценки фармакокинетики и иммуногенности препаратов бевацизумаба. В исследование были включены ..."
 
Vol 11, No 3 (2022) Development and Validation of HPLC-UV Method for the Determination of Favipiravir in Human Plasma Abstract  PDF (Eng)  similar documents
T. N. Komarov, P. K. Karnakova, O. A. Archakova, D. S. Shchelgacheva, N. S. Bagaeva, I. E. Shohin, K. Ya. Zaslavskaya, P. A. Bely
"... использованием ультрафиолетового детектора (ВЭЖХ-УФ) для дальнейшего изучения фармакокинетики. Материалы и ..."
 
Vol 12, No 2 (2023) Simultaneous Determination of Nirmatrelvir and Ritonavir in Human Plasma by HPLC-MS/MS Abstract  PDF (Eng)  similar documents
T. N. Komarov, P. K. Karnakova, O. A. Archakova, D. S. Shchelgacheva, N. S. Bagaeva, I. E. Shohin, K. Ya. Zaslavskaya, P. A. Bely
"... / МС) для дальнейшего изучения фармакокинетики. Материалы и методы. Определение нирматрелвира и ..."
 
Vol 13, No 1 (2024) Development and Validation of an HPLC-MS/MS Method for Quantification of Apixaban in Human Plasma Abstract  PDF (Eng)  similar documents
U. D. Filonova, P. K. Karnakova, K. K. Karnakova, M. O. Popova, A. A. Popova, O. A. Archakova, T. N. Komarov, I. E. Shohin
 
Vol 11, No 2 (2022) Development and Validation of the HPLC Method for Quantification of the Innovative Drug DD217, Factor Xa Inhibitor, in Rat Plasma for a Pharmacokinetic Study Abstract  PDF (Rus)  similar documents
N. S. Dubovik, D. F. Guranda, G. V. Ramenskaya, D. G. Tovbin, D. N. Tarasov, A. Yu. Savchenko, V. S. Arnautov
"... for the pharmaceutical market. One of such drugs is N-(5-chloropyridine-2-yl)-2-({4-[ethanimidoyl(methyl)benzoyl}amino)-5 ..."
 
Vol 8, No 3 (2019) Study of Lercanidipine Drug Release from Medicine in Combination with Ramipril in vitro and in vivo Abstract  PDF (Rus)  similar documents
A. A. Shadrin, D. Y. Ivkin, E. V. Flisyuk, I. E. Smekhova, G. A. Plisko, A. A. Karpov, E. D. Semivelichenko
"... комбинациям препаратов в одной таблетке. Изучение фармакокинетики лекарственных веществ и учет их ..."
 
Vol 9, No 2 (2020) Results of the Estimation of Biosimilarity of RinLiz® (LLC «GEROPHARM», Russia) and Humalog® (Lilly France, France) Using the Method of the Hyperinsulinemic Eulygemic Clamp on Healthy Voluntary Abstract  PDF (Rus)  similar documents
A. Yu. Mayorov, I. A. Fedotov, R. V. Drai, O. I. Avdeeva, I. E. Makarenko
"... клинических исследований (КИ) биоаналогов инсулина входят исследования фармакологии: фармакокинетика (ФК ..."
 
Vol 13, No 3 (2024) Development and validation of the method of quantification of 5-[5-(trifluoromethyl)-1,2-oxazole-3-yl]-furan-2-sulfonamide and its metabolites in laboratory animal plasma Abstract  PDF (Rus)  similar documents
I. I. Yaichkov, M. K. Korsakov, A. A. Shetnev, N. N. Volkhin, S. S. Petukhov
"... determination of this compound and its N-hydroxy- and N-acetyl metabolites in the plasma of laboratory animals ..."
 
Vol 12, No 1 (2023) Simultaneous Determination of Major Molnupiravir Metabolite (β-D-N4-hydroxycytidine) and Favipiravir in Human Plasma by HPLC-MS/MS Abstract  PDF (Eng)  similar documents
T. N. Komarov, P. K. Karnakova, O. A. Archakova, D. S. Shchelgacheva, N. S. Bagaeva, I. E. Shohin, K. Ya. Zaslavskaya, P. A. Bely
"... chromatography – tandem mass spectrometry (HPLC-MS/MS) method for the simultaneous determination of β-D-N4 ..."
 
Vol 9, No 4 (2020) Indolo[2,3-a]carbazole Derivatives with Antitumor Activity and Instrumental Methods for Their Investigation (Review) Abstract  PDF (Rus)  similar documents
D. A. Kozin, Z. S. Shprakh, V. Yu. Reshetnyak, O. V. Nesterova, I. N. Avertseva, G. M. Rodionova
"... . Yu., Nesterova O. V., Avertseva I. N., Rodionova G. M. Indolo[2,3-a]carbazole derivatives with ..."
 
Vol 13, No 1 (2024) Development and Validation of an HPLC-MS/MS Method for the Quantitative Determination of Etmaben in Human Blood Plasma Abstract  PDF (Rus)  similar documents
P. K. Karnakova, T. N. Komarov, O. A. Archakova, D. Yu. Ivkin, E. S. Vetrova, I. I. Terninko, I. E. Shohin, I. A. Narkevich
"... preparation: precipitation with acetonitrile. Internal standard: promethazine. Column: Luna C18, 100 Å, 50 × 2 ..."
 
Vol 9, No 3 (2020) Dypeptydylpeptidase IV Activity Ingibition after Oral Administration to Rabbits of Strongylocentrotus Droebahiensis Gonads Extract as Possible Biomarker of Pharmakokinetics Abstract  PDF (Rus)  similar documents
V. M. Kosman, N. M. Faustova, I. N. Urakova, M. N. Karlina, V. G. Makarov
"... ). Традиционные подходы к изучению фармакокинетики, основанные на применении хроматографических методов, зачастую ..."
 
Vol 14, No 2 (2025) The excretion study of a new derivative of 4,5-dihydroisoxazole-5-carboxamide Abstract  PDF (Rus)  similar documents
I. I. Yaichkov, M. K. Korsakov, N. N. Volkhin, V. E. Zaykova, O. E. Lasaraynz
"... -yl)-N-[4-methoxy-3-(trifluoromethyl)phenyl]-4,5-dihydro-1,2-oxazole-5-carboxamide (R004 ..."
 
Vol 8, No 3 (2019) Development and Validation of HPLC-MS/MS Method for Busereline Quantitation in Animal Blood Plasma Abstract  PDF (Rus)  similar documents
E. N. Fisher, E. S. Melnikov, I. Е. Shohin
"... определения бусерелина в плазме крови с целью исследования фармакокинетики. ..."
 
Vol 9, No 2 (2020) The Study of Pharmacokinetics Parameters of Morphine Hydrochloride, Long-acting Tablets in Cancer Patients with Severe Chronic Pain Syndrome Abstract  PDF (Rus)  similar documents
E. A. Ezhova, I. G. Kotelnikova, A. V. Teteneva, D. V. Butuzova, K. F. Tetenev
"... сильной интенсивности. Материалы и методы. Для анализа фармакокинетики исследуемого препарата после ..."
 
Vol 8, No 3 (2019) Evaluation of Pharmacokinetical Parameters of Phenol, a Component of Antiseptic Dorogov's stimulator 3 Fraction Paste Abstract  PDF (Rus)  similar documents
V. I. Nozdrin, G. A. Piavchenko, M. E. Ivanova, K. S. Guzev, S. L. Kuznetsov
"... Дорогова 3 фракции был получен более полувека назад, до настоящего времени сведения о фармакокинетике ..."
 
Vol 13, No 4 (2024) Pharmacokinetic study of a new 4,5-dihydroisoxazole-5-carboxamide derivative in rats Abstract  PDF (Rus)  similar documents
I. I. Yaichkov, M. K. Korsakov, N. N. Volkhin, S. S. Petukhov, A. N. Tyushina, V. E. Zaykova, O. E. Lasaraynz
"... Introduction. 3-(2-butyl-5-chloro-1H-imidazole-4-yl)-N-[4-methoxy-3-(trifluoromethyl)phenyl]-4 ..."
 
Vol 13, No 4 (2024) Phase I pharmacokinetic study of etmaben, a malonic acid derivative Abstract  PDF (Rus)  similar documents
P. K. Karnakova, K. K. Karnakova, T. N. Komarov, N. S. Bagaevа, M. O. Popova, D. Yu. Ivkin, O. A. Archakova, I. E. Shohin, I. A. Narkevich
"... «Этмабен» находится на фазе I клинических исследований (КИ), ранее его фармакокинетика у человека не ..."
 
Vol 10, No 2 (2021) Comparative Pharmacokinetics Study of 1-[2-(2-benzoylphenoxy)ethyl]-6-methyluracil Substance and its Solid Dispersion Systems on Rabbits Abstract  PDF (Rus)  similar documents
V. M. Kosman, D. V. Demchenko, E. A. Jain (Korsakova), V. G. Makarov, V. Yu. Balabanyan
"... Введение. Изучение фармакокинетики лекарственных веществ и оценка их фармакокинетических ..."
 
Vol 13, No 4 (2024) Pharmacokinetics of a new drug based on polysaccharide from acorus calamus in an experiment on laboratory animals Abstract  PDF (Rus)  similar documents
S. V. Krivoshchekov, E. A. Yanovskaya, R. V. Gurto, O. S. Bryushinina, D. A. Isakov, A. V. Zykova, Yu. G. Zyuz’kova, A. M. Guryev, V. V. Udut, M. V. Belousov
"... образования галактуроновой кислоты. Результаты и обсуждения. Изучена фармакокинетика нового лекарственного ..."
 
1 - 36 of 36 Items

Search tips:

  • Search terms are case-insensitive
  • Common words are ignored
  • By default articles containing any term in the query are returned (i.e., OR is implied)
  • Make sure that a word exists in an article by prefixing it with +; e.g., +journal +access scholarly academic
  • Combine multiple words with AND to find articles containing all terms; e.g., education AND research
  • Exclude a word by prefixing it with - or NOT; e.g., online -politics or online NOT politics
  • Search for an exact phrase by putting it in quotes; e.g., "open access publishing". Hint: Quoting Chinese or Japanese words will help you to find exact word matches in mixed-language fields, e.g. "中国".
  • Use parentheses to create more complex queries; e.g., archive ((journal AND conference) NOT theses)